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RecruitingNCT06382012AFTR NV RCTUpdated May 18, 2026

Antiemetic Fosaprepitant To Remedy Nausea and Vomiting

A Phase 2/3 interventional study of Fosaprepitant 150 mg and Ondansetron 4 mg in Nausea and Vomiting, Nausea and Vomiting, sponsored by Montefiore Medical Center. Recruiting at 1 site in United States. Open to participants aged 18 Years and older. Per ClinicalTrials.gov, last updated 2026-05-18.

Sponsored by Montefiore Medical Center · Phase 2/3, Interventional, and Treatment

Phase
Phase 2/3
Study type
Interventional
Enrollment
200
Allocation
Randomized
Ages
18 Years and older
Sex
All
01

Study summary

The study team proposes a randomized, double-blind, RCT to address the following goal: to determine the relative efficacy and adverse event profile of fosaprepitant compared to the standard of care antiemetic ondansetron. Fosaprepitant and its active metabolite aprepitant are a relatively new class of antiemetic that exclusively acts in the central nervous system by blocking neurokinin (NK-1) which is a key signaling molecule in the centrally mediated aspects of the vomiting reflex. Currently, fosaprepitant and aprepitant both have only two United Stated Food and Drug Administration (USFDA) approved indications for nausea and vomiting: chemotherapy-induced and postoperative. Neurokinin inhibitors are highly effective and generally well-tolerated. Therefore, this class of medication may be a more appropriate medication for the millions of patients with nausea and vomiting that seek care in EDs. Intravenous fosaprepitant is converted to the active metabolite aprepitant on the order of minutes and is significantly cheaper to procure at this time. The outcome for the efficacy analysis will be no need for additional medication to treat nausea and vomiting within 2 hours of investigational medication administration. The primary outcome for the tolerability analysis will be the development of any new symptom within 2 hours of medication administration.

Read the detailed description

Nausea and vomiting (NV) are common and interrelated conditions. Approximately 50% of adults experience nausea in a given year while 30% of adults experience vomiting over the same period. Of this population of symptomatic individuals with NV, 25% of patients seek care in any healthcare delivery setting. Health Care Utilization Project (HCUP) data indicates that nearly 9.0 million patients seek care for NV in emergency departments (EDs) each year in the United States.

Antiemetics are used to treat NV. Antiemetics currently utilized in the emergency department setting for NV do not always work on the first dose and have a plethora of side effects because of their peripheral mechanism of action outside of the vomiting reflex pathway in the central nervous system. These medications include ondansetron, promethazine, metoclopramide, olanzapine, haloperidol. Chief among these side effects is alteration of an aspect cardiac electrical signaling called the QT segment which represents the duration of ventricular contraction and relaxation. The QT segment is prolonged with commonly used antiemetics which can often be a prelude to cardiac dysrhythmias that are associated with mortality. As a result, patients with NV often have long length-of-stay (LOS) involving supportive care with intravenous fluids or empiric treatment with medications that can potentiate development of cardiac dysrhythmias. This is a problem in busy emergency departments (EDs) struggling to accelerate patient throughput in order to appropriately keep up with patient volume in an under-supplied hospital bed environment nationally.

Fosaprepitant and its active metabolite aprepitant are a relatively new class of antiemetic that exclusively acts in the central nervous system by blocking neurokinin (NK-1) which is a key signaling molecule in the centrally mediated aspects of the vomiting reflex. Currently, fosaprepitant and aprepitant both have only two United Stated Food and Drug Administration (USFDA) approved indications for nausea and vomiting: chemotherapy-induced and postoperative. Neurokinin inhibitors are highly effective and generally well-tolerated. Therefore, this class of medication may be a more appropriate medication for the millions of patients with nausea and vomiting that seek care in EDs. Intravenous fosaprepitant is converted to the active metabolite aprepitant on the order of minutes and is significantly cheaper to procure at this time.

02

Conditions studied

  • Nausea and Vomiting
  • Nausea
  • Vomiting

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Keywords

  • Fosaprepitant
  • Vomiting
  • Randomized Control Trial
  • Ondansetron
  • Adults
03

Who can participate

Ages eligible
18 Years and older
Sexes eligible
All
Accepts healthy volunteers
No

Inclusion criteria

  • Adults at least 18 years old
  • Present to an emergency department (ED) for nausea and/or vomiting as defined by the International Classification of Diseases (ICD-10), or identified by treating clinician
  • Following the approval of a protocol amendment, study patients who have received an antiemetic and remain persistently nauseated after 2 hours will be eligible to participate in the study

Exclusion criteria

Exclusion Criteria:

  • Pregnancy, desiring pregnancy, or lactating
  • Antiemetic medication use less than 2 hours prior to screening
  • Bradycardia (heart rate less than 60 bpm heart rate)
  • Prolonged QTc (>480ms)
  • Not conversant in English or Spanish
  • Altered mental status
  • Dementia
  • Lack of phone for follow-up communication
04

Study design

Phase
Phase 2 / Phase 3
Primary purpose
Treatment
Allocation
Randomized
Intervention model
Parallel assignment
Masking
Quadruple (Participant, Care provider, Investigator, Outcomes assessor)
Enrollment
200 participants (estimated)

Study arms

  • Experimental
    Investigational Intervention

    Fosaprepitant 150mg IV administered over 15 minutes

    Drug: Fosaprepitant 150 mg

  • Active comparator
    Standard-of-Care Intervention

    Ondansetron 4mg IV administered over 15 minutes

    Drug: Ondansetron 4 mg

Interventions

  • DrugFosaprepitant 150 mg

    Fosaprepitant 150mg IV administered over 15 minutes

  • DrugOndansetron 4 mg

    Ondansetron 4mg IV administered over 15 minutes

05

What researchers measure

Primary outcomes

  1. Relief from NV

    Relief from nausea and vomiting will be determined by the intensity of nausea reported by participants following administration of antiemetic. Intensity of nausea will be reported as either "None," "Mild," "Moderate," or "Severe." Relief of nausea and vomiting requires a patient to present with a nausea intensity of either "Severe" or "Moderate," which is then reduced by treatment to at least "Mild" or "None," within two hours of medication administration, without the use or rescue medication. The number/percentage of participants who achieve relief from NV will be summarized by study arm.

    Time frame: Within 2 hours of medication administration

  2. Occurrence of any treatment-related adverse event

    The primary safety/tolerability outcome for this study is the occurrence of any treatment related adverse event (TRAE) at 2 hours of medication administration. TRAEs - not including underlying pathology causing NV - and including, but not limited to: appendicitis, small bowel obstruction, constipation, gastroparesis, gastroenteritis, gastritis, will be summarized by study arm

    Time frame: 2 hours following medication administration

  3. Requirement for additional medication

    Requirement of any additional medication specifically for treatment of NV at 2 hours of medication administration; the use of rescue medications to treat persistent NV, or other medications such as additional doses or use of adjunct medications will be recorded. The number/percentage of patients who require additional medication will be summarized by study arm.

    Time frame: 2 hours following medication administration

Secondary outcomes

  1. Freedom from nausea and vomiting (NV)

    Freedom from nausea and vomiting (NV) will be determined by the intensity of nausea reported by participants following administration of antiemetic. Intensity of nausea will be reported as either "None," "Mild," "Moderate," or "Severe." Sustained freedom from nausea and vomiting requires a patient to present with a nausea intensity of either "Severe" or "Moderate," which is then reduced by treatment to "None" within two hours of medication administration. The number/percentage of patients with freedom from nausea/vomiting (NV) will be measured every 15 minutes for the first 2 hours. The number/percentage of patients with freedom from NV at 2 hours will be summarized by study arm.

    Time frame: 2 hours following medication administration

  2. Sustained Relief from nausea and vomiting (NV) (at 24 hours)

    The number/percentage of patients demonstrating relief from nausea/vomiting (NV) will be measured every 15 minutes for the first 2 hours (for assessment of the primary outcome), then during every hour up to the end of the follow up period at 24 hours. Relief from NV is defined as achieving a level of relief of either "Mild" or None" at 2 hours and maintaining that level of "Mild" or "None" for the entire 24-hour period following medication administration, without use of rescue medication. The number/percentage of participants who achieve relief from NV will be summarized by study arm.

    Time frame: At 24-hours following medication administration

  3. Sustained NV Freedom (at 24 hours)

    Sustained freedom from nausea and vomiting (NV) will be determined by the intensity of nausea reported by participants following administration of antiemetic. Intensity of nausea will be reported as either "None," "Mild," "Moderate," or "Severe." Sustained freedom from nausea and vomiting requires a patient to present with a nausea intensity of either "Severe" or "Moderate," which is then reduced by treatment to "None" within two hours of medication administration (corresponding secondary outcome), and maintained at this level (i.e., "None") for the entire 24-hour follow-up period, without the use or rescue medication. The number/percentage of participants who achieve sustained freedom from NV will be summarized by study arm.

    Time frame: At 24- hours following medication administration

  4. Disposition Plan

    A disposition determination plan will be documented at 4 hours. Patients will be categorized as either having been either "admitted," "discharged," or status "yet to be determined." Categorical data will be summarized by study arm.

    Time frame: 4 hours following medication administration

  5. Patient Medication Preference for subsequent episode of NV

    Medication preference will be assessed based on patient's preference for receiving the same antiemetic medication as administered for a subsequent episode of nausea and vomiting. Binary ("Yes" for having the same medication administered, "No" for request of a different medication) responses of patient preference will be summarized by study arm.

    Time frame: 24 hours following medication administration

  6. Emergency Department (ED) Length of Stay (LOS)

    ED LOS will be defined as the interval of time from initial presentation to final disposition in the ED, will be determined. Mean LOS results will be summarized by study arm.

    Time frame: From initial presentation to disposition in ED, approximately 4 hours

Other outcomes

  1. Severity of Nausea

    Mean severity of nausea scores will be evaluated and summarized based on a visual analogue scale from 0 to 100 (0 = no nausea, 100 = worst nausea possible) such that higher scores are associated with more severe nausea. Results will be summarized by study arm.

    Time frame: 24 hours (measured every 15 minutes for the first 2 hours, then hourly after that until disposition; reassessed at 24 hours)

  2. Functional disability

    Patient reported functional disability will be assessed. Functional disability will be categorized as either "Severe," "Moderate," "Mild," or "Not impaired." Categorical variables will be summarized by study arm using descriptive statistics.

    Time frame: 24 hours (assessed prior to receiving intervention, at 2 hour point after receiving intervention, and 24 hours after intervention)

  3. Number of Vomiting Episodes

    The mean number of vomiting episodes per patient will be determined and summarized by study arm.

    Time frame: 24 hours following medication administration

  4. Need for rescue antiemetic medication

    Binary outcome for needing or not needing additional dosing of antiemetic medication to treat nausea will be determined. Results will be summarized by study arm.

    Time frame: 2 hours (assessed at the 2 hour mark after administration of the intervention)

  5. Number of Patients Requiring Hospitalization

    The number/percentage of patients who require hospitalization within 24 hours due to NV symptoms will be determined. Results will be summarized by study arm.

    Time frame: 24 hours

  6. Fluid Treatment

    The percentage of patients treated with IV fluids will be determined. Results will be summarized by study arm.

    Time frame: 4 hours

  7. Mean Fluid Volume

    The mean per patient volume of IV fluids administered will be summarized by study arm.

    Time frame: 4 hours

  8. QTc Interval (QT interval corrected for heart rate)

    Mean QTc durations, as calculated from ECG readings administered prior to receiving intervention and at disposition, will be determined. Prolonged QT interval is commonly associated with antiemetics and can often be a prelude to cardiac dysrhythmias associated with mortality. Mean QTc durations will be summarized by study arm.

    Time frame: Prior to Intervention and at disposition, approximately 2 hours

  9. Revisit Rate

    Revisit rate will be assessed as the number/percentage of participants requiring a revisit to the Emergency department for NV. Results will be summarized by study arm.

    Time frame: 24 hours

06

Study locations

1 of 1 sites recruiting
  • Montefiore Medical Center (Montefiore and Weiler EDs)
    The Bronx, New York 10467, United States
    Recruiting
07

References and documents

Publications

  • Mechanisms and Control of Emesis: A Satellite Symposium of the European Neuroscience Association: Proceedings of an International Meeting Held in Marseille (France), 4-7 September 1992. John Libbey Eurotext
  • Singh P, Yoon SS, Kuo B. Nausea: a review of pathophysiology and therapeutics. Ther Adv Gastroenterol. 2016 Jan;9(1):98-112. doi: 10.1177/1756283X15618131. PubMed 26770271 ↗
  • Healthcare Cost and Utilization Project (HCUP) Statistical Briefs [Internet]. Rockville (MD): Agency for Healthcare Research and Quality (US); 2006 Feb-. Available from http://www.ncbi.nlm.nih.gov/books/NBK52651/ PubMed 21413206 ↗
  • Pourmand A, Mazer-Amirshahi M, Chistov S, Sabha Y, Vukomanovic D, Almulhim M. Emergency department approach to QTc prolongation. Am J Emerg Med. 2017 Dec;35(12):1928-1933. doi: 10.1016/j.ajem.2017.08.044. Epub 2017 Aug 24. PubMed 28855066 ↗
  • Franklin BJ, Vakili S, Huckman RS, Hosein S, Falk N, Cheng K, Murray M, Harris S, Morris CA, Goralnick E. The Inpatient Discharge Lounge as a Potential Mechanism to Mitigate Emergency Department Boarding and Crowding. Ann Emerg Med. 2020 Jun;75(6):704-714. doi: 10.1016/j.annemergmed.2019.12.002. Epub 2020 Jan 23. PubMed 31983501 ↗
  • Aapro M, Carides A, Rapoport BL, Schmoll HJ, Zhang L, Warr D. Aprepitant and fosaprepitant: a 10-year review of efficacy and safety. Oncologist. 2015 Apr;20(4):450-8. doi: 10.1634/theoncologist.2014-0229. Epub 2015 Mar 20. PubMed 25795636 ↗
  • Langford P, Chrisp P. Fosaprepitant and aprepitant: an update of the evidence for their place in the prevention of chemotherapy-induced nausea and vomiting. Core Evid. 2010 Oct 21;5:77-90. doi: 10.2147/ce.s6012. PubMed 21042544 ↗
  • Furyk JS, Meek RA, Egerton-Warburton D. Drugs for the treatment of nausea and vomiting in adults in the emergency department setting. Cochrane Database Syst Rev. 2015 Sep 28;2015(9):CD010106. doi: 10.1002/14651858.CD010106.pub2. PubMed 26411330 ↗
  • Yang Y, Yang N, Wu L, Ouyang Q, Fang J, Li J, Liao W, Cai K, Huang J, Li J, Zhang Y, Wang X, Zhang H, Xu N, Zhao Q, Hu X, Li W, Zhong W, Zhong D, Cheng G, Ye S, Zhong M, Wang D, Liu H, Zheng J, Liu X, Xu H, Zhang L. Safety and efficacy of aprepitant as mono and combination therapy for the prevention of emetogenic chemotherapy-induced nausea and vomiting: post-marketing surveillance in China. Chin Clin Oncol. 2020 Oct;9(5):68. doi: 10.21037/cco-20-160. PubMed 33161724 ↗
  • Tramer MR, Phillips C, Reynolds DJ, McQuay HJ, Moore RA. Cost-effectiveness of ondansetron for postoperative nausea and vomiting. Anaesthesia. 1999 Mar;54(3):226-34. doi: 10.1046/j.1365-2044.1999.00704.x. PubMed 10364857 ↗

Individual participant data

Plan to share: No

08

Registry details

Key details

Study ID
NCT06382012
Lead sponsor
Montefiore Medical Center
Responsible party
Sponsor
First posted
Apr 24, 2024
Start date
Nov 13, 2024
Primary completion
Mar 2027 (estimated)
Completion
Mar 2027 (estimated)
Last update
May 18, 2026

Study contacts

Mustfa K Manzur, MD MPH MS
Contact
mmanzur@montefiore.org
718-920-6626
Benjamin W Friedman, MD MS
principal investigator · Montefiore Medical Center

Oversight

Data monitoring committee
Yes
FDA-regulated drug
Yes
FDA-regulated device
No
View the source record on ClinicalTrials.gov ↗

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