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CompletedNCT04983238Updated Jan 5, 2024

Evaluation of Safety and Efficacy of Sodium Thiosulfate (BYON5667) Eye Drops to Reduce Ocular Toxicity in Cancer Patients Treated With SYD985

A Phase 1/2 interventional study of BYON5667 & SYD985 and Placebo & SYD985 in Metastatic Breast Cancer, sponsored by Byondis B.V.. Completed at 10 sites in 3 countries. Open to female participants aged 18 Years and older. Per ClinicalTrials.gov, last updated 2024-01-05.

Sponsored by Byondis B.V. · Phase 1/2, Interventional, and Prevention

Phase
Phase 1/2
Study type
Interventional
Enrollment
48
Allocation
Randomized
Ages
18 Years and older
Sex
Female
01

Study summary

This multicenter, randomized, double-blind, placebo-controlled trial with a single arm run-in period is to evaluate the safety and efficacy of sodium thiosulfate (BYON5667) eye drops to reduce ocular toxicity in cancer patients treated with the antibody-drug conjugate (ADC) SYD985

Read the detailed description

This multicenter trial has a single arm run-in period followed by a randomized, placebo-controlled, double-blind comparative part. In the single arm part of the trial, patients with HER2-expressing locally advanced or metastatic solid tumours will be enrolled and treated with the antibody-drug conjugate (ADC) SYD985 once every 3 weeks until disease progression or unacceptable toxicity. All patients will receive concomitant BYON5667 eye drops. When the primary safety and efficacy analysis of the BYON5667 eye drops at Day 63 is favorable, the trial may continue to the comparative part in which patients with locally advanced or metastatic HER2-positive breast cancer will be treated with SYD985. Patients will be randomly assigned (1:1) to receive BYON5667 or placebo eye drops.

02

Conditions studied

  • Metastatic Breast Cancer
03

Who can participate

Ages eligible
18 Years and older
Sexes eligible
Female
Accepts healthy volunteers
No

Eligibility criteria

Main Inclusion Criteria:

  1. Male or female, age ≥18 years at the time of signing first informed consent;
  2. Patient with histologically-confirmed, unresectable locally advanced or metastatic cancer with the following restriction:

    Single arm part: patient with solid tumours of any origin (excluding gastric tumours and adenocarcinomas of the gastroesophageal junction) who has progressed on standard therapy or for whom no standard therapy exists; Randomized part: patient with breast cancer who had either progression during or after at least two human epidermal growth factor receptor 2 (HER2)-targeting treatment regimens for locally advanced or metastatic disease, or progression during or after [ado-]trastuzumab emtansine treatment for locally advanced or metastatic disease;

  3. HER2 tumour status as determined by a local laboratory using immunohistochemistry (IHC) and/or in situ hybridization (ISH):

    Single arm part: at least IHC 1+; Randomized part: IHC 3+ and/or ISH positive;

  4. Eastern Cooperative Oncology Group (ECOG) performance status ≤ 1;
  5. Patient should refrain from wearing any kind of contact lenses during trial treatment;
  6. Adequate organ function

Main Exclusion Criteria:

  1. Current or previous use of prohibited medication as listed in the protocol
  2. History of infusion-related reactions and/or hypersensitivity to trastuzumab containing treatment or excipients of the trial treatments which led to permanent discontinuation of the treatment;
  3. History or presence of keratitis;
  4. Left ventricular ejection fraction (LVEF) \< 50%, or a history of clinically significant decrease in LVEF during previous trastuzumab containing treatment leading to permanent discontinuation of treatment;
  5. History or presence of idiopathic pulmonary fibrosis, organizing pneumonia (e.g. bronchiolitis obliterans), drug-induced or idiopathic pneumonitis, or evidence of active pneumonitis on screening chest CT scan;
  6. History or presence of clinically significant cardiovascular disease;
  7. Severe, uncontrolled systemic disease;
  8. Symptomatic brain metastases, brain metastases requiring steroids to manage symptoms, or treatment for brain metastases within 8 weeks.
04

Study design

Phase
Phase 1 / Phase 2
Primary purpose
Prevention
Allocation
Randomized
Intervention model
Parallel assignment
Masking
Triple (Participant, Care provider, Investigator)
Enrollment
48 participants (actual)

Study arms

  • Experimental
    BYON5667 & SYD985

    BYON5667 eye drops should be self-administered daily during waking hours. SYD985, every 3 weeks (Q3W)

    Drug: BYON5667 & SYD985

  • Placebo comparator
    Placebo & SYD985

    Placebo eye drops should be self-administered daily during waking hours. SYD985, every 3 weeks (Q3W)

    Drug: Placebo & SYD985

Interventions

  • DrugBYON5667 & SYD985

    Ocular administration: BYON5667, Intravenous administration: SYD985

    Also known as: BYON5667: sodium thiosulfate, SYD985: (vic-)trastuzumab duocarmazine

  • DrugPlacebo & SYD985

    Ocular administration: Placebo, Intravenous administration: SYD985

    Also known as: SYD985: (vic-)trastuzumab duocarmazine

05

What researchers measure

Primary outcomes

  1. Efficacy of BYON5667 eye drops by assessing the percentage of patients with SYD985-related ocular adverse events Grade >=1 at Day 63

    Percentage of patients with SYD985-related ocular toxicity Grade ≥1 at Day 63

    Time frame: 63 days

Secondary outcomes

  1. Ocular toxicity

    Percentage of patients with SYD985-related ocular toxicity of different grades at Day 63 or Day 126

    Time frame: Day 63 or Day 126

  2. Tolerability of BYON5667 eye drops by means of Eye Drop Tolerability questionnaire scores

    Tolerability of BYON5667 eye drops Questionnaire includes 5 questions with score of 0 (no discomfort) to 10 (most imaginable discomfort)

    Time frame: Up to 2 years

  3. National Eye Institute Visual Function Questionnaire (NEI VFQ-25) scores

    Self-reported validated questionnaire including 25 questions with scores of 1 to maximum 6, from best/worst to worst/best depending on the question

    Time frame: Up to 2 years

  4. SYD985-related ocular adverse events (AE)

    Time to first SYD985-related ocular AE

    Time frame: Up to 2 years

  5. Discontinuation due to SYD985-related ocular toxicity

    Percentage of patients discontinued due to SYD985-related ocular toxicity

    Time frame: Up to 2 years

  6. Efficacy of SYD985 by assessing the objective response rate (ORR)

    Efficacy of SYD985

    Time frame: Up to 2 years

  7. Efficacy of SYD985 by assessing the progression-free survival (PFS)

    Efficacy of SYD985

    Time frame: Up to 2 years

  8. Efficacy of SYD985 by assessing the overall survival

    Efficacy of SYD985

    Time frame: Up to 2 years

  9. Safety of SYD985 by assessing incidence and severity of treatment-emergent drug-related adverse events

    Safety of SYD985

    Time frame: Up to 2 years

06

Study locations

10 sites
  • University Hospital Antwerp
    Antwerp, 2650, Belgium
  • UZ Leuven
    Leuven, 3000, Belgium
  • Institut Bergonié
    Bordeaux, 33076, France
  • Centre Oscar Lambret
    Lille, 59020, France
  • Hôpital Saint Louis
    Paris, 75475, France
  • Vall d' Hebron
    Barcelona, 8035, Spain
  • ICO I'Hospitalet - Hospital Duran i Reynals
    L'Hospitalet De Llobregat, 8908, Spain
  • Hospital Universitari Arnau de Vilanova
    Lleida, 25198, Spain
  • START Madrid HU Fundacion Jimenez Diaz
    Madrid, 28040, Spain
  • START Madrid HU HM Sanchinarro
    Madrid, 28050, Spain
07

References and documents

Individual participant data

Plan to share: No

No publications or documents are linked to this record.

08

Registry details

Key details

Study ID
NCT04983238
Lead sponsor
Byondis B.V.
Responsible party
Sponsor
First posted
Jul 30, 2021
Start date
Jan 10, 2022
Primary completion
Apr 19, 2023
Completion
Jun 26, 2023
Last update
Jan 5, 2024

Study contacts

Ellen Mommers, PhD
study director · Byondis B.V., The Netherlands

Oversight

Data monitoring committee
Yes
FDA-regulated drug
No
FDA-regulated device
No
View the source record on ClinicalTrials.gov ↗

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