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CompletedNCT06488664Updated Sep 21, 2026

An Efficacy and Safety Study of GNR-068 (Ustekinumab Biosimilar) and Stelara® in the Treatment of Patients With Moderate to Severe Plaque Psoriasis

A Phase 3 interventional study of GNR-068 and Stelara® in Plaque Psoriasis, sponsored by AO GENERIUM. Completed at 34 sites in Russia. Open to participants aged 18 Years to 75 Years. Per ClinicalTrials.gov, last updated 2026-09-21.

Sponsored by AO GENERIUM · Phase 3, Interventional, and Treatment

Phase
Phase 3
Study type
Interventional
Enrollment
422
Allocation
Randomized
Ages
18 Years to 75 Years
Sex
All
01

Study summary

This is a randomized single-blind comparative parallel group efficacy and safety study of ustekinumab biosimilar GNR-068 (45 mg) and reference product Stelara® (45 mg) in the treatment of patients with moderate and severe forms of plaque psoriasis. Participants received a subcutaneous dose of ustekinumab 45 mg (GNR-068 or Stelara®) at weeks 0 and 4 weeks then every 12 weeks thereafter until week 28 and then all patients receive GNR-068 45 mg. For patients with partially respond to the initial regimen the regimen can be adjusted.

Read the detailed description

The drug GNR-068 (INN: ustekinumab) is being developed as a biosimilar to the drug Stelara®, solution for subcutaneous administration (Silag AG, Switzerland).

Preclinical studies and early phase clinical studies suggest that interleukins-12 (IL-12) and -23 (IL-23), two molecules that are part of the communication network in the immune system, may play an important role in psoriasis. Ustekinumab is a monoclonal antibody directed against IL-12 and IL-23. This is a randomized, single blind, parallel-group, multicenter study to determine the effectiveness and safety of ustekinumab biosimilar GNR-068 administered subcutaneously as compared with Stelara® in patients with moderate to severe plaque-type psoriasis. Patients receive GNR-068 45 mg or Stelara 45 mg administered subcutaneously at weeks 0 and 4 weeks then every 12 weeks thereafter until week 28, thereafter until week 52 all patients receive GNR-068. For patients who partially respond to the initial regimen, the dose can be adjusted to 90 mg and then the interval can be adjusted to every 8 weeks. The study included a screening period, comparative treatment period, non-comparative treatment period, follow up period. Allocation of patients to treatment groups was carried out by randomization in a ratio of 1:1. 422 patients (211 to each study groups) were randomized.

02

Conditions studied

  • Plaque Psoriasis

Keywords

  • ustekinumab
  • humanized monoclonal antibodies
  • safety
  • plaque psoriasis
  • equivalence
  • biosimilar
  • PASI (Psoriasis Area and Severity Index)
  • BSA (Body Surface Area)
  • DLQI (Dermatological Life Quality Index)
  • PGA (Physician's Global Assessment)
  • immunogenicity
03

Who can participate

Ages eligible
18 Years to 75 Years
Sexes eligible
All
Accepts healthy volunteers
No

Inclusion criteria

  • Written informed consent to participate in the study.
  • Men and women 18-75 years of age, inclusive, at the time of signing the informed consent form.
  • Patients diagnosed with plaque psoriasis at least 6 months before screening:

    1. Moderate or severe form of the disease, which is defined as: PASI index ≥12, body surface area (BSA) affected by plaque psoriasis, ≥10%, PGA scale score ≥3 (on a scale from 0 to 4).
    2. Presence of indications for systemic therapy, defined as inadequate control of the disease against the background of: local treatment (including local glucocorticosteroids) and/or phototherapy and/or lack of clinical effect from the use of other systemic methods.
    3. It is acceptable to carry out basic therapy for psoriatic arthritis at a stable dose for ≥ 4 weeks before screening: prednisolone at a dose of ≤10 mg per day, NSAIDs, methotrexate at a dose of ≤15 mg per week, sulfasalazine at a dose of 2.0 g per day.
  • Body weight less than 100 kg.
  • If it is necessary to take drugs that worsen the course of psoriasis (beta blockers, calcium channel blockers, lithium drugs, etc.): a stable dose of these drugs for ≥ 4 weeks before randomization.
  • Consent of women of childbearing age, women in menopause lasting less than 2 years and male patients to comply with adequate methods of contraception throughout the study and for 3 months after the end of ustekinumab therapy.
  • Patients should not be donors of blood or its components 30 days before inclusion in the study and not become donors of blood or its components throughout the study and for 3 months after its completion.

Exclusion criteria

Exclusion Criteria:

  • Types of psoriasis other than plaque, except for concomitant psoriatic arthritis.
  • History of therapy with ustekinumab or any therapy aimed at IL-12 or IL-23 (briakinumab, guselkumab, tildrakizumab).
  • Therapy with TNF-alpha inhibitors or any other genetically engineered biological drugs within 3 months before randomization.
  • Conducting other systemic therapies (including cyclosporine, acitretin, methotrexate, UV and PUVA therapy) within 1 month before randomization.
  • Treatment with leflunomide for 6 months before randomization.
  • Spread of the inflammatory process involving the gastrointestinal tract (inflammatory bowel diseases), the organ of vision (uveitis, iridocyclitis), musculoskeletal structures (high activity of psoriatic arthritis, osteoarthritis, uncontrolled against the background of basic therapy (clause 3 Inclusion criteria) ).
  • Major surgery (including joint surgery) within 8 weeks before the start of the study or elective surgery within 6 months after the start of the study.
  • A history of an adverse drug reaction to any of the components of the study drug or a reference drug.
  • Immunization with any live or live attenuated vaccine within 1 month before the first dose of the study drug or comparator drug.
  • A history of a disease associated with the accumulation of immune complexes that may distort the assessment of the effectiveness of ustekinumab therapy (including serum sickness, systemic lupus erythematosus, rheumatoid arthritis, polymyositis, scleroderma, Sjogren's syndrome, vasculitis, cryoglobulinemia).
  • Concomitant diseases and conditions that, in the opinion of the Investigator and/or Sponsor, jeopardize the safety of the patient during participation in the study, or which will influence the analysis of safety data.
  • Active systemic infection (bacterial, viral or fungal) within 14 days before signing the informed consent.
  • Pregnancy or breastfeeding.
  • History of tuberculosis, positive/doubtful result of screening for tuberculosis infection (tuberculosis allergen test or IGRA test or fluorography results). Inclusion of such patients is possible if effective specific treatment for tuberculosis infection has been carried out and there is a conclusion from a phthisiatrician about the possibility of ustekinumab therapy.
  • Participation in clinical trials of drugs less than 5 half-lives of the study drug before signing the informed consent.
  • Positive test for hepatitis B or C, HIV or syphilis.
  • Unwillingness or inability to comply with the recommendations prescribed by this protocol.
  • Identification during screening of other diseases/conditions not listed above that, in the opinion of the physician-researcher, prevent the inclusion of the patient in the study.
04

Study design

Phase
Phase 3
Primary purpose
Treatment
Allocation
Randomized
Intervention model
Parallel assignment
Masking
Single (Participant)
Enrollment
422 participants (actual)

Study arms

  • Experimental
    GNR-068 (JSC "GENERIUM", Russia)

    Test drug

    Biological: GNR-068

  • Active comparator
    Stelara® (manufacturer Silag AG, Switzerland)

    reference drug

    Biological: Stelara®

Interventions

  • BiologicalGNR-068

    GNR-068 was administered subcutaneously at weeks 0 and 4 weeks then every 12 weeks thereafter until week 52.

    Also known as: ustekinumab biosimilar

  • BiologicalStelara®

    Stelara® was administered subcutaneously at weeks 0 and 4 weeks then every 12 weeks thereafter until week 28 and then all patients receive GNR-068 45 mg until week 52.

    Also known as: ustekinumab

05

What researchers measure

Primary outcomes

  1. The proportion of subjects with Psoriasis Area and Severity Index (PASI) Score of 75 Percent or Above

    PASI is a widely used tool for the measurement of severity of psoriasis. This is a test of how bad a person's psoriasis is. The scale combines redness, scaling, and thickness, as well as overall body involvement to determine the PASI score. The scale ranges from 0 (best) to 72 (worst).

    Time frame: Week 12

Secondary outcomes

  1. The proportion of patients achieving PASI50/75/90/100

    PASI is a widely used tool for the measurement of severity of psoriasis. This is a test of how bad a person's psoriasis is. The scale combines redness, scaling, and thickness, as well as overall body involvement to determine the PASI score. The scale ranges from 0 (best) to 72 (worst).

    Time frame: Week 60

  2. Time to reach PASI50, PASI75, PASI90, PASI100

    PASI is a widely used tool for the measurement of severity of psoriasis. This is a test of how bad a person's psoriasis is. The scale combines redness, scaling, and thickness, as well as overall body involvement to determine the PASI score. The scale ranges from 0 (best) to 72 (worst).

    Time frame: Week 60

  3. Area under the curve (AUC) of PASI

    PASI is a widely used tool for the measurement of severity of psoriasis. This is a test of how bad a person's psoriasis is. The scale combines redness, scaling, and thickness, as well as overall body involvement to determine the PASI score. The scale ranges from 0 (best) to 72 (worst).

    Time frame: Week 60

  4. The proportion of partial responders (ie, patients achieving ≥50% but <75% improvement in PASI compared to baseline)

    PASI is a widely used tool for the measurement of severity of psoriasis. This is a test of how bad a person's psoriasis is. The scale combines redness, scaling, and thickness, as well as overall body involvement to determine the PASI score. The scale ranges from 0 (best) to 72 (worst).

    Time frame: Week 60

  5. Changes in the BSA index

    Using the BSA (Body Surface Area) index, the surface area of the skin affected by psoriasis is assessed. BSA is measured in %. To determine the area of psoriatic skin lesions the "palm" rule is applicable. On the scalp, the affected area the size of one palm is assumed to be 10%, the torso - 3.3%, the upper extremities - 5%, the lower extremities - 2.5% of the area of the anatomical region of the body. To calculate the total BSA, each reported percentage must be multiplied by the corresponding factor of the corresponding body region (head = 0.1, torso = 0.3, upper extremities = 0.2, lower extremities = 0.4). The resulting four percentage values (percentage of skin affected by psoriasis on the scalp, upper extremities, trunk, and lower extremities) will be summed to estimate the BSA index.

    Time frame: Week 60

  6. Changes in PGA

    The PGA is 7-point scale used in clinical trials of various diseases. In this the physician checks the state of the disease and gives them score from 0 (clear) to 5 (severe).

    Time frame: Week 60

  7. Changes in the intensity of itching on the visual analogue scale (VAS)

    The intensity of itching is carried out at all visits using a visual analogue scale (VAS), where the left end of the line is 0 = no itching, the right end of the line is 10 = intense itching

    Time frame: Week 60

  8. Changes in quality of life, assessed using the Dermatology Life Quality Index (DLQI)

    The DLQI is a 10-item questionnaire, that in addition to evaluating overall quality of life, can be used to assess 6 different aspects that may affect quality of life: symptoms and feelings, daily activities, leisure, work or school performance, personal relationships, and treatment. Scores range from 0 (no impairment in quality of life) to 30 (most impairment in quality of life).

    Time frame: Week 60

  9. The proportion of patients who dropped out of the study due to lack of sufficient therapeutic response

    Treatment failure is assessed as no effect within 28 weeks (PASI response \<50%)

    Time frame: Week 60

06

Study locations

34 sites
  • Federal State Budgetary Educational Institution of Higher Education "Altai State Medical University" of the Ministry of Health of the Russian Federation
    Barnaul, Barnaul 656038, Russia
  • State budgetary healthcare institution "Chelyabinsk Regional Clinical Dermatovenerological Dispensary"
    Chelyabinsk, Chelyabinsk Oblast 454048, Russia
  • Limited Liability Company "Ecology of Health"
    Chelyabinsk, Chelyabinsk Oblast 454126, Russia
  • State budgetary institution of the Sverdlovsk region "Ural Research Institute of Dermatovenereology and Immunopathology"
    Yekaterinburg, Ekaterinburg 620076, Russia
  • Limited Liability Company "Alliance Biomedical - Ural Group"
    Izhevsk, Izhevsk 426061, Russia
  • Federal State Budgetary Educational Institution of Higher Education "Kirov State Medical University" of the Ministry of Health of the Russian Federation (FSBEI HE Kirov State Medical University of the Ministry of Health of Russia))
    Kirov, Kirov Oblast 610027, Russia
  • Limited Liability Company "Available Polyclinic"
    Murino, Leningradskaya Oblast' 188678, Russia
  • State health care institution "Regional Dermatovenerological Dispensary"
    Lipetsk, Lipetsk Oblast 398005, Russia
  • Limited Liability Company "OLLA-MED"
    Moscow, Moscow 105554, Russia
  • Federal State Budgetary Institution "Research Institute of Rheumatology named after V.A. Nasonova"
    Moscow, Moscow 115522, Russia
  • Limited Liability Company "Firma ORIS"
    Moscow, Moscow 117321, Russia
  • State budgetary healthcare institution of the city of Moscow "Moscow Scientific and Practical Center of Dermatovenereology and Cosmetology of the Moscow Health Department"
    Moscow, Moscow 119071, Russia
  • Federal State Budgetary Educational Institution of Higher Education "Russian University of Medicine" of the Ministry of Health of the Russian Federation (FSBEI HE "Russian University of Medicine" of the Ministry of Health of Russia)
    Moscow, Moscow 127006, Russia
  • State budgetary healthcare institution of the Moscow region "Moscow Regional Research Clinical Institute named after M.F. Vladimirsky"
    Moscow, Moscow 129110, Russia
  • Limited Liability Company "Family Clinic No. 4"
    Korolyov, Moscow Oblast 141060, Russia
  • Limited Liability Company "Medical Center "Healthy Family"
    Novosibirsk, Novosibirsk Oblast 630099, Russia
  • Federal State Budgetary Educational Institution of Higher Education Orenburg State Medical University of the Ministry of Health of Russia
    Orenburg, Orenburg Oblast 460018, Russia
  • State budgetary institution of the Ryazan region "Regional clinical dermatovenerological dispensary"
    Ryazan, Ryazan Oblast 390046, Russia
  • Limited Liability Company "Clinic of Skin Diseases Pierre Wolkenstein"
    Saint Petersburg, Sankt-Peterburg 191123, Russia
  • Limited Liability Company "International Medical Center"
    Saint Petersburg, Sankt-Peterburg 191123, Russia
  • Limited Liability Company "Medical Technologies" LLC "Medical Technologies"
    Saint Petersburg, Sankt-Peterburg 192148, Russia
  • Limited Liability Company "Health Energy"
    Saint Petersburg, Sankt-Peterburg 194156, Russia
  • Limited Liability Company "Interleukin"
    Saint Petersburg, Sankt-Peterburg 194214, Russia
  • Limited Liability Company "Institute of Medical Research"
    Saint Petersburg, Sankt-Peterburg 196084, Russia
  • Limited Liability Company "Research Center Eco-Safety"
    Saint Petersburg, Sankt-Peterburg 196143, Russia
  • Limited Liability Company "PiterKlinika"
    Saint Petersburg, Sankt-Peterburg 196158, Russia
  • Limited Liability Company "ArsVite North-West"
    Saint Petersburg, Sankt-Peterburg 196191, Russia
  • Limited Liability Company "Curator"
    Saint Petersburg, Sankt-Peterburg 196240, Russia
  • Private medical institution "Euromedservice"
    Saint Petersburg, Sankt-Peterburg 196603, Russia
  • Limited Liability Company "MEDINET"
    Saint Petersburg, Sankt-Peterburg 197136, Russia
  • Limited Liability Company "SB Clinic of Cosmetology"
    Saratov, Saratov Oblast 410012, Russia
  • Regional state budgetary healthcare institution "Smolensk Dermatovenerological Dispensary"
    Smolensk, Smolensk Oblast 214031, Russia
  • Limited Liability Company Medical Center "Azbuka Health"
    Kazan', Tatarstan Republic 420111, Russia
  • State Budgetary Healthcare Institution Ulyanovsk area Clinical Hospital
    Ulyanovsk, Ulyanovsk Oblast 432063, Russia
07

References and documents

Individual participant data

Plan to share: No

No publications or documents are linked to this record.

08

Registry details

Key details

Study ID
NCT06488664
Lead sponsor
AO GENERIUM
Responsible party
Sponsor
First posted
Jul 5, 2024
Start date
Jul 25, 2023
Primary completion
Apr 30, 2025
Completion
Nov 26, 2025
Last update
Sep 21, 2026

Study contacts

Oksana A. Markova, MD
study chair · JSC GENERIUM

Oversight

Data monitoring committee
No
FDA-regulated drug
No
FDA-regulated device
No
View the source record on ClinicalTrials.gov ↗

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