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RecruitingNCT05785065SSc-mILDUpdated Sep 29, 2026

Mycophenolate Mofetil in Systemic Sclerosis With Subclinical Interstitial Lung Disease

A Phase 2 interventional study of Mycophenolate Mofetil and Placebo in Systemic Sclerosis With Lung Involvement, Systemic Sclerosis and Interstitial Lung Disease, sponsored by Centre hospitalier de l'Université de Montréal (CHUM). Recruiting at 3 sites in Canada. Open to participants aged 18 Years and older. Per ClinicalTrials.gov, last updated 2026-09-29.

Sponsored by Centre hospitalier de l'Université de Montréal (CHUM) · Phase 2, Interventional, and Other

Phase
Phase 2
Study type
Interventional
Enrollment
35
Allocation
Randomized
Ages
18 Years and older
Sex
All
01

Study summary

The goal of this pilot study is to assess the feasibility of a larger study on the efficacy of mycophenolate mofetil in people diagnosed with systemic sclerosis with mild lung involvement. Participants will be recruited over 12 months at 3 academic centers and assigned randomly to receive either mycophenolate mofetil or placebo, a look-alike substance that contains no active drug, for 96 weeks.

Read the detailed description

Background: Systemic sclerosis (SSc, scleroderma) is a rare but life-threatening systemic autoimmune disease characterized by microvasculopathy, serum autoantibodies, inflammation and fibrosis of the skin and internal organs. Early rapidly progressive SSc remains the most lethal autoimmune rheumatic disease, with over 60% mortality at 5 years in high-risk patients. Interstitial lung disease (ILD) is the leading cause of SSc-related mortality and affects over half of SSc patients. SSc-ILD is currently treated with immunosuppressive and anti-fibrotic drugs, with the first-line treatment being mycophenolate mofetil (MMF), although treatments have modest benefits when initiated in advanced stages of disease. Emerging data suggest that earlier treatment, when lung function is still normal despite evidence of ILD on computed tomography scan ("subclinical SSc-ILD"), may lead to improved outcomes, suggesting a window of treatment opportunity.

Research Aims: The goal of the proposed pilot RCT is to establish the feasibility of a phase III RCT that will assess the efficacy of MMF in subclinical SSc-ILD. Specifically, we aim to:

  1. Determine the rate of patient recruitment at three centers over one year, and identify barriers and solutions to recruitment;
  2. Determine the proportion of participants receiving the allocated treatment and with complete primary efficacy outcome data at 48 and 96 weeks; and
  3. Generate preliminary data on clinical efficacy outcomes that will contribute information to the analysis of the phase III trial through a Bayesian inference framework.

Methods: Participants will be adults with SSc, ILD diagnosed within the past 3 years and a normal forced vital capacity (≥ 80%). Participants will be recruited over 12 months at 3 academic centers affiliated to the Canadian Scleroderma Research Group. Eligible participants will be assigned using stratified randomization to receive either MMF (up to 2 grams daily) or placebo for 96 weeks. The primary feasibility outcome will be the rate of recruitment per site over 12 months. A Bayesian approach will be used to estimate the probability of reaching the target sample size based on observed recruitment rates, with decision rules to continue, adapt, or stop the trial. Data collected on the primary clinical efficacy outcome (annual rate of decline in forced vital capacity over 96 weeks) will be used to inform the analysis of the phase III trial (as an informative prior) through a Bayesian inference framework.

02

Conditions studied

  • Systemic Sclerosis With Lung Involvement
  • Systemic Sclerosis
  • Interstitial Lung Disease

Keywords

  • Systemic sclerosis
  • Mycophenolate mofetil
  • Interstitial lung disease
03

Who can participate

Ages eligible
18 Years and older
Sexes eligible
All
Accepts healthy volunteers
No

Inclusion criteria

  1. Able and willing to provide informed consent and adhere to study protocol;
  2. Women and men of all race/ethnicity, aged 18 years and older;
  3. SSc based on 2013 ACR-EULAR classification criteria;
  4. Presence of interstitial lung disease on HRCT scan, obtained within 12 months before screening, that shows fibrosis affecting less than 20% of the lungs, as confirmed by an expert radiologist;
  5. Diagnosis of ILD within 7 years before screening;
  6. Forced vital capacity of 80% predicted and above, on pulmonary function tests obtained within 6 months before screening;
  7. Able to communicate in French or English;

Exclusion criteria

Exclusion Criteria:

  1. Progressive pulmonary fibrosis, defined as at least two of three criteria (worsening symptoms, radiological progression, and physiological progression) occurring within the past year with no alternative explanation, as defined by the 2022 ATS/ERS/JRS/ALAT Clinical Practice Guideline;
  2. Use of medications with putative lung disease-modifying properties:

    1. Current use of MMF, mycophenolic acid, azathioprine, calcineurin inhibitors (e.g. tacrolimus, cyclosporin A), tocilizumab, nintedanib, pirfenidone or corticosteroids (Prednisone equivalent dose >10 mg/day) at time of screening
    2. Cyclophosphamide within one year prior to screening
    3. Rituximab within 6 months prior to screening
    4. Cell therapies (including stem cell transplantation) within one year prior to screening
  3. Current use of other biological, targeted synthetic or investigational products with immunosuppressive effects (e.g. TNF inhibitors, abatacept, tofacitinib) at time of screening
  4. Any contraindication to MMF, including:

    1. Pregnancy and/or breastfeeding
    2. Female of childbearing potential not using reliable method of contraception
    3. Persistent leucopenia (white blood cell count \<3.0 x103/μL)
    4. Persistent thrombocytopenia (platelet count \<100 x103/μL)
    5. Persistent anemia (hemoglobin \<100 g/L)
    6. Baseline liver enzymes (alanine transaminase (ALT) or aspartate transaminase (AST)) or bilirubin >1.5 times the upper limit of normal, other than due to Gilbert's disease
    7. Uncontrolled congestive heart failure
    8. Active infection (lung or elsewhere)
    9. Active solid or hematological malignancy (other than basal cell cancer of the skin or cervical carcinoma in situ removed entirely by biopsy)
    10. Active peptic ulcer disease
    11. Other serious concomitant medical illness, unreliability or drug abuse that might compromise the patient's ability to safely take MMF
    12. Use of drugs or products with significant interactions with MMF
04

Study design

Phase
Phase 2
Primary purpose
Other
Allocation
Randomized
Intervention model
Parallel assignment
Masking
Quadruple (Participant, Care provider, Investigator, Outcomes assessor)
Enrollment
35 participants (estimated)

Study arms

  • Experimental
    Mycophenolate mofetil

    2 to 4 capsules of mycophenolate mofetil twice daily.

    Drug: Mycophenolate Mofetil

  • Placebo comparator
    Placebo

    2 to 4 capsules of placebo twice daily.

    Other: Placebo

Interventions

  • DrugMycophenolate Mofetil

    The participant will receive 500 mg to 1000 mg twice daily of mycophenolate mofetil administered orally for 96 weeks. The dose scheduling will be as follow: Weeks 1 and 2: 500 mg twice a day Weeks 3 and 4: 750 mg twice a day Weeks 5 to 96: 1000 mg twice a day

  • OtherPlacebo

    The participant will receive 500 mg to 1000 mg twice daily of placebo administered orally for 96 weeks. The dose scheduling will be as follow: Weeks 1 and 2: 500 mg twice a day Weeks 3 and 4: 750 mg twice a day Weeks 5 to 96: 1000 mg twice a day

05

What researchers measure

Primary outcomes

  1. Total number of potentially eligible patients identified per site

    Time frame: Over one year

  2. Proportion of potentially eligible patients who provide consent per site

    Time frame: Over one year

  3. Proportion of consented participants who meet the eligibility criteria per site

    Time frame: Over one year

  4. Monthly rate of randomized participants per site

    Time frame: Over one year

  5. Adherence to treatment as assessed by Participant Dosing Diaries

    Time frame: From the first dose to the last dose taken for each participant, up to 96 weeks

  6. Drug adherence rate as assessed by Pharmacy Accountability Logs

    Time frame: From the first dose to the last dose taken for each participant, up to 96 weeks

  7. Adherence to the study protocol as assessed by the number of protocol deviations

    Time frame: Over total study period (up to 96 weeks per participant)

  8. Proportion of participants intolerant to the study drug who discontinue trial treatment

    Time frame: Over total study period (up to 96 weeks per participant)

  9. Proportion of participants receiving the allocated treatment at 48 weeks

    Time frame: At 48 weeks

  10. Proportion of participants receiving the allocated treatment at 96 weeks

    Time frame: At 96 weeks

  11. Proportion of participants with complete primary efficacy outcome data at 48 weeks

    Time frame: At 48 weeks

  12. Proportion of participants with complete primary efficacy outcome data at 96 weeks

    Time frame: At 96 weeks

  13. Proportion of participants lost to follow-up

    Time frame: Over total study period (up to 96 weeks per participant)

Secondary outcomes

  1. Frequency of treatment-related adverse events

    Incidence and severity of AEs, with severity determined according to National Cancer Institute Common Terminology Criteria for Adverse Events, Version 5.0 (NCI CTCAE v5.0)

    Time frame: Over total study period (up to 96 weeks per participant)

Other outcomes

  1. Annual rate of decline in percent (%) predicted forced vital capacity (FVC) over 48 weeks

    Time frame: Over 48 weeks

  2. Annual rate of decline in percent (%) predicted forced vital capacity (FVC) over 96 weeks

    Time frame: Over 96 weeks

  3. Proportion of participants having clinically meaningful progression

    Clinically meaningful progression defined by the Outcome Measures in Rheumatology (OMERACT) for connective tissue disease-associated interstitial lung diseases (CTD-ILD) (defined as a ≥10% relative decline in FVC from baseline, or a ≥5% to \<10% relative decline in FVC associated with a ≥15% relative decline in diffusion capacity \[DLCO\])

    Time frame: Over total study period (up to 96 weeks per participant)

  4. Time to clinically meaningful progression

    Clinically meaningful progression as defined by Outcome Measures in Rheumatology (OMERACT) for connective tissue disease- associated interstitial lung diseases (CTD-ILD) (defined as a ≥10% relative decline in FVC from baseline, or a ≥5% to \<10% relative decline in FVC associated with a ≥15% relative decline in diffusion capacity \[DLCO\])

    Time frame: Over total study period (up to 96 weeks per participant)

  5. Proportion of participants having an absolute decrease in FVC of at least 3.3% predicted

    An absolute decrease in FVC of at least 3.3% predicted was proposed as the minimal clinically important difference estimate for worsening of FVC in patients with SSc-ILD.

    Time frame: Over total study period (up to 96 weeks per participant)

  6. Time to an absolute decrease in FVC of at least 3.3% predicted

    An absolute decrease in FVC of at least 3.3% predicted was proposed as the minimal clinically important difference estimate for worsening of FVC in patients with SSc-ILD.

    Time frame: Over total study period (up to 96 weeks per participant)

  7. Proportion of participants having progressive pulmonary fibrosis

    Progressive pulmonary fibrosis defined by 2022 ATS/ERS/JRS/ALAT guidelines

    Time frame: Over total study period (up to 96 weeks per participant)

  8. Time to progressive pulmonary fibrosis

    Progressive pulmonary fibrosis defined by 2022 ATS/ERS/JRS/ALAT guidelines

    Time frame: Over total study period (up to 96 weeks per participant)

  9. Annual rate of decline in percent (%) predicted total lung capacity over 48 weeks

    Time frame: Over 48 weeks

  10. Annual rate of decline in percent (%) predicted total lung capacity over 96 weeks

    Time frame: Over 96 weeks

  11. Annual rate of decline in percent (%) predicted diffusion capacity for carbon monoxide (DLCO) over 48 weeks

    Time frame: Over 48 weeks

  12. Annual rate of decline in percent (%) predicted DLCO over 96 weeks

    Time frame: Over 96 weeks

  13. Change from baseline in percent (%) extent of ILD, ground-glass opacities, reticular infiltrates and honeycombing, and in pulmonary vessel volume at 48 weeks

    Measured on high-resolution computed tomography chest scan using automated lung texture analysis

    Time frame: At 48 weeks

  14. Change from baseline in percent (%) extent of ILD, ground-glass opacities, reticular infiltrates and honeycombing, and in pulmonary vessel volume at 96 weeks

    Measured on high-resolution computed tomography chest scan using automated lung texture analysis

    Time frame: At 96 weeks

  15. Change from baseline in St-George Respiratory Questionnaire at 48 weeks

    Scores range from 0 to 100, with higher scores indicating more limitations.

    Time frame: At 48 weeks

  16. Change from baseline in St-George Respiratory Questionnaire at 96 weeks

    Scores range from 0 to 100, with higher scores indicating more limitations.

    Time frame: At 96 weeks

  17. Change from baseline in Leicester Cough Questionnaire at 48 weeks

    Scores (total) range from 3 to 21, with higher scores indicating less limitations.

    Time frame: At 48 weeks

  18. Change from baseline in Leicester Cough Questionnaire at 96 weeks

    Scores (total) range from 3 to 21, with higher scores indicating less limitations.

    Time frame: At 96 weeks

  19. Change from baseline in health assessment questionnaire modified for scleroderma at 48 weeks

    The SHAQ consists of the Health assessment questionnaire (HAQ) and visual analogue scales for pain, patient global assessment, vascular, digital ulcers, lung involvement and gastrointestinal involvement. Scores range from 0 to 3, with higher scores indicating more limitations.

    Time frame: At 48 weeks

  20. Change from baseline in health assessment questionnaire modified for scleroderma at 96 weeks

    The SHAQ consists of the Health assessment questionnaire (HAQ) and visual analogue scales for pain, patient global assessment, vascular, digital ulcers, lung involvement and gastrointestinal involvement. Scores range from 0 to 3, with higher scores indicating more limitations.

    Time frame: At 96 weeks

  21. Change from baseline in 36-items short form survey (SF-36) at 48 weeks

    Eight scales with scores range from 0 to 100, with higher scores indicating less limitations.

    Time frame: At 48 weeks

  22. Change from baseline in 36-items short form survey (SF-36) at 96 weeks

    Eight scales with scores ranging from 0 to 100, with higher scores indicating less limitations.

    Time frame: At 96 weeks

  23. Change from baseline in EuroQoL five dimensions (EQ-5D-5L) at 48 weeks

    The EQ-5D-5L questionnaire possesses 5 levels for each of the five dimensions. The five dimensions are mobility, self-care, usual activities, pain/discomfort, and anxiety/depression, with the following possible five responses: no problems, slight problems, moderate problems, severe problems, unable to/extreme problems. Scores are converted into an index value ranging from 0 to 1, with higher scores indicating better health state.

    Time frame: At 48 weeks

  24. Change from baseline in EuroQoL five dimensions (EQ-5D-5L) at 96 weeks

    The EQ-5D-5L questionnaire possesses 5 levels for each of the five dimensions. The five dimensions are mobility, self-care, usual activities, pain/discomfort, and anxiety/depression, with the following possible five responses: no problems, slight problems, moderate problems, severe problems, unable to/extreme problems. Scores are converted into an index value ranging from 0 to 1, with higher scores indicating better health state.

    Time frame: At 96 weeks

  25. Change from baseline in patient global assessment at 48 weeks

    Visual analogue scale from 0 to 10, with higher scores indicating worse disease.

    Time frame: At 48 weeks

  26. Change from baseline in patient global assessment at 96 weeks

    Visual analogue scale from 0 to 10, with higher scores indicating worse disease.

    Time frame: At 96 weeks

  27. Change from baseline in physician global assessment at 48 weeks

    Visual analogue scale from 0 to 10, with higher scores indicating worse disease.

    Time frame: At 48 weeks

  28. Change from baseline in physician global assessment at 96 weeks

    Visual analogue scale from 0 to 10, with higher scores indicating worse disease.

    Time frame: At 96 weeks

  29. Change from baseline in 6-minute walk oxygen saturation at 48 weeks

    Oxygen saturation at nadir during the 6-minute walk test

    Time frame: At 48 weeks

  30. Change from baseline in 6-minute walk oxygen desaturation at 96 weeks

    Oxygen saturation at nadir during the 6-minute walk test

    Time frame: At 96 weeks

  31. Change from baseline in modified Rodnan skin score (mRSS) at 48 weeks

    Scores range from 0 to 51, with higher scores indicating more skin involvement.

    Time frame: At 48 weeks

  32. Change from baseline in modified Rodnan skin score (mRSS) at 96 weeks

    Scores range from 0 to 51, with higher scores indicating more skin involvement.

    Time frame: At 96 weeks

  33. Change from baseline in nailfold capillary density at 48 weeks

    Mean number of capillaries per mm

    Time frame: At 48 weeks

  34. Change from baseline in nailfold capillary density at 96 weeks

    Mean number of capillaries per mm

    Time frame: At 96 weeks

  35. Change from baseline in nailfold capillaroscopy abnormalities and patterns at 48 weeks

    Ectasias/megacapillaries are scored using a semi-quantitative scale (0 = no, 1 = ≤33%, 2= 33-66%, and 3 = ≥66% abnormalities/linear mm)

    Time frame: At 48 weeks

  36. Change from baseline in nailfold capillaroscopy abnormalities and patterns at 96 weeks

    Ectasias/megacapillaries are scored using a semi-quantitative scale (0 = no, 1 = ≤33%, 2= 33-66%, and 3 = ≥66% abnormalities/linear mm)

    Time frame: At 96 weeks

  37. Change from baseline in quantitative SSc autoantibody titers at 48 weeks

    Time frame: At 48 weeks

  38. Change from baseline in quantitative SSc autoantibody titers at 96 weeks

    Time frame: At 96 weeks

  39. Change from baseline in Krebs von Lungen 6 (KL-6) titers at 48 weeks

    Time frame: At 48 weeks

  40. Change from baseline in Krebs von Lungen 6 (KL-6) titers at 96 weeks

    Time frame: At 96 weeks

06

Study locations

1 of 3 sites recruiting
  • Centre hospitalier de l'Université de Montréal (CHUM)
    Montreal, Quebec H2X 3E4, Canada
    Recruiting
  • Jewish General Hospital - CIUSSS-COMTL
    Montreal, Quebec H3T 1E2, Canada
    • Marie Hudson, MD · Contact
    • Marie Hudson, MD · Principal investigator
    Not yet recruiting
  • Institut Universitaire de Cardiologie et Pneumologie de Québec
    Québec, Quebec, Canada
    Not yet recruiting
07

Registry details

Key details

Study ID
NCT05785065
Lead sponsor
Centre hospitalier de l'Université de Montréal (CHUM)
Collaborators
McGill University, University of Calgary, Jewish General Hospital, Canadian Institutes of Health Research (CIHR), Sclérodermie Québec, Institut universitaire de cardiologie et de pneumologie de Québec, University Laval
Responsible party
Sponsor
First posted
Mar 27, 2023
Start date
Aug 29, 2024
Primary completion
Dec 2026 (estimated)
Completion
Dec 2028 (estimated)
Last update
Sep 29, 2026

Study contacts

Sabrina Hoa, MD MSc
Contact
sabrina.anh-tu.hoa.med@ssss.gouv.qc.ca
514-890-8000
Unité d'innovation thérapeutique, CHUM
Contact
uit.eligibilite.chum@ssss.gouv.qc.ca
Sabrina Hoa, MD
principal investigator · Centre hospitalier de l'Université de Montréal (CHUM)

Oversight

Data monitoring committee
No
FDA-regulated drug
No
FDA-regulated device
No
View the source record on ClinicalTrials.gov ↗

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