CClinicalTrials.gg
Not yet recruitingNCT07750041Updated Aug 6, 2026

A Phase Ib/II Study of SYS6090 Combination Therapy in Advanced Colorectal Cancer

A Phase 1/2 interventional study of SYS6090 (Fixed Dose Level A) + bevacizumab and SYS6090 (Fixed Dose Level B ) + bevacizumab in Unresectable Advanced or Metastatic Colorectal Cancer, sponsored by CSPC Megalith Biopharmaceutical Co.,Ltd.. Not yet recruiting at 1 site in China. Open to participants aged 18 Years and older. Per ClinicalTrials.gov, last updated 2026-08-06.

Sponsored by CSPC Megalith Biopharmaceutical Co.,Ltd. · Phase 1/2, Interventional, and Treatment

Phase
Phase 1/2
Study type
Interventional
Enrollment
260
Allocation
Randomized
Ages
18 Years and older
Sex
All
01

Study summary

This study constitutes an open-label, multi-cohort, multi-center Phase Ib/II clinical study, developed to assess the safety, tolerability, and therapeutic efficacy of SYS6090 injection when administered in combination with bevacizumab, or in triple combination with bevacizumab and chemotherapy, among patients diagnosed with advanced colorectal cancer.

02

Conditions studied

  • Unresectable Advanced or Metastatic Colorectal Cancer
03

Who can participate

Ages eligible
18 Years and older
Sexes eligible
All
Accepts healthy volunteers
No

*Eligibility Criteria:

Inclusion criteria

Inclusion Criteria:

  1. Subjects must be ≥18 years of age.
  2. Histologically or cytologically confirmed unresectable advanced or metastatic colorectal cancer with pMMR/MSS status, assigned to corresponding cohorts as follows:

    Cohort 1 (2L/3L) of Phase Ib \& Phase II: Subjects must have disease progression after no more than 2 lines of standard systemic therapy (prior regimens must contain fluoropyrimidine-, oxaliplatin-, and irinotecan-based chemotherapy); tumor tissue confirmed as pMMR by IHC or MSS by NGS/PCR; Cohort 2 (1L) of Phase Ib \& Phase II: Subjects have received no prior systemic anti-tumor therapy for advanced disease; tumor tissue confirmed as pMMR by IHC or MSS by NGS/PCR.

  3. At least one extracranial measurable lesion at baseline according to RECIST 1.1 criteria.
  4. Eastern Cooperative Oncology Group performance status of 0 or 1.
  5. Expected survival ≥ 3 months.
  6. Has protocol-defined adequate organ and bone marrow function.

Exclusion criteria

Exclusion Criteria:

  1. Subjects with clinically active central nervous system metastases;
  2. with a history of other primary malignant tumors within 5 years before administration;
  3. Subjects assigned to Cohort 1 who have received prior regorafenib treatment.;
  4. Prior documented interstitial lung disease (ILD)/ pneumonitis that required steroids, current ILD/ pneumonitis, or suspected ILD/ pneumonitis that cannot be ruled out by imaging at screening;
  5. Uncontrolled or significant cardiovascular disease;
  6. Clinically uncontrolled pleural effusion, ascites or pericardial effusion;
  7. Has unresolved toxicities from previous anticancer therapy, defined as toxicities not yet resolved to Grade ≤ 1 or baseline .
04

Study design

Phase
Phase 1 / Phase 2
Primary purpose
Treatment
Allocation
Randomized
Intervention model
Parallel assignment
Masking
None (open label)
Enrollment
260 participants (estimated)

Study arms

  • Experimental
    Ib-Randomized Arm 1

    Enrolled Subjects will be randomized to receive SYS6090 at the fixed dose level A in combination with bevacizumab. The exact dose magnitude and administration frequency of SYS6090 are temporarily undisclosed to protect pending patent information, with full dosing details archived in platform backend for regulatory review only.

    Drug: SYS6090 (Fixed Dose Level A) + bevacizumab

  • Experimental
    Ib-Randomized Arm 2

    Enrolled Subjects will be randomized to receive SYS6090 at the fixed dose level B in combination with bevacizumab. The exact dose magnitude and administration frequency of SYS6090 are temporarily undisclosed to protect pending patent information, with full dosing details archived in platform backend for regulatory review only.

    Drug: SYS6090 (Fixed Dose Level B ) + bevacizumab

  • Experimental
    II-Cohort 1- Randomized Arm A

    Enrolled Subjects will be randomized to receive SYS6090 at RP2D combined with bevacizumab and mFOLFOX6

    Drug: SYS6090 RP2D + bevacizumab +mFOLFOX6

  • Experimental
    II-Cohort 1- Randomized Arm B

    Enrolled Subjects will be randomized to receive SYS6090 at RP2D combined with bevacizumab

    Drug: SYS6090 RP2D + bevacizumab

  • Experimental
    II-Cohort 1- Randomized Arm C

    Enrolled Subjects will be randomized to receive regorafenib

    Drug: Regorafenib

  • Experimental
    II-Cohort 2- Randomized Arm D

    Enrolled Subjects will be randomized to receive SYS6090 at RP2D combined with bevacizumab and FOLFOXIRI

    Drug: SYS6090 PR2D+ bevacizumab + FOLFOXIRI

  • Active comparator
    II-Cohort 2- Randomized Arm E

    Enrolled Subjects will be randomized to receive bevacizumab combined with FOLFOXIRI

    Drug: bevacizumab + FOLFOXIRI

Interventions

  • DrugSYS6090 (Fixed Dose Level A) + bevacizumab

    Participants will receive intravenous SYS6090 at fixed dose level A combined with intravenous bevacizumab, administered per cycle schedule specified in study protocol, for advanced/palliative unresectable pMMR/MSS colorectal cancer.

  • DrugSYS6090 (Fixed Dose Level B ) + bevacizumab

    Participants will receive intravenous SYS6090 at fixed dose level B plus intravenous bevacizumab per protocol-defined cycle schedule for unresectable advanced pMMR/MSS colorectal cancer.

  • DrugSYS6090 RP2D + bevacizumab +mFOLFOX6

    Participants will receive intravenous SYS6090 at RP2D plus intravenous bevacizumab combined with standard mFOLFOX6 chemotherapy regimen (oxaliplatin, leucovorin, fluorouracil), administered per protocol-defined cycle schedule for unresectable advanced pMMR/MSS colorectal cancer.

  • DrugSYS6090 RP2D + bevacizumab

    Participants will receive intravenous SYS6090 at RP2D plus intravenous bevacizumab, administered per protocol-defined cycle schedule for unresectable advanced pMMR/MSS colorectal cancer.

  • DrugRegorafenib

    Oral regorafenib monotherapy as standard control for metastatic pMMR/MSS colorectal cancer.

  • DrugSYS6090 PR2D+ bevacizumab + FOLFOXIRI

    Participants will receive intravenous SYS6090at RP2D plus intravenous bevacizumab combined with FOLFOXIRI triple chemotherapy (oxaliplatin, irinotecan, leucovorin, fluorouracil) per study cycle schedule for metastatic pMMR/MSS colorectal cancer.

  • Drugbevacizumab + FOLFOXIRI

    Participants will receive intravenous bevacizumab combined with FOLFOXIRI triple chemotherapy (oxaliplatin, irinotecan, leucovorin, fluorouracil) per study cycle schedule for metastatic pMMR/MSS colorectal cancer.

05

What researchers measure

Primary outcomes

  1. Recommended Phase 2 Dose (RP2D), Safety and Tolerability

    RP2D of SYS6090 combination therapy,Safety and tolerability are evaluated via incidence and severity of all Adverse Events (AEs) and Serious Adverse Events (SAEs) graded per NCI-CTCAE version 6.0, including abnormal laboratory tests, ECG parameters and vital signs from screening through end of safety follow-up.

    Time frame: up to approximately 3 years after the first enrollment

  2. Objective Response Rate (ORR) assessed per RECIST v1.1

    ORR per Response Evaluation Criteria in Solid Tumors version 1.1 (RECIST 1.1) assessed by investigator was defined as the percentage of participants with at least one visit confirmed complete response (CR) or partial response (PR), for all cohorts in Phase Ib and Cohort 1 of Phase II expansion stage.

    Time frame: up to approximately 3 years after the first enrollment

  3. Progression-Free Survival (PFS) assessed per RECIST v1.1

    PFS per Response Evaluation Criteria in Solid Tumors version 1.1 (RECIST 1.1) assessed by investigator was defined as the time from the date of randomization or first study treatment until the date of confirmed progressive disease (PD), or death by any cause in the absence of progression, regardless of whether the participant withdrew from study therapy or received another anticancer therapy prior to progression, for Cohort 2 of Phase II expansion stage.

    Time frame: up to approximately 3 years after the first enrollment

06

Study locations

1 site
07

Registry details

Key details

Study ID
NCT07750041
Lead sponsor
CSPC Megalith Biopharmaceutical Co.,Ltd.
Responsible party
Sponsor
First posted
Aug 6, 2026
Start date
Aug 30, 2026 (estimated)
Primary completion
Dec 31, 2027 (estimated)
Completion
Aug 30, 2029 (estimated)
Last update
Aug 6, 2026

Study contacts

Clinical Trials Information Group officer
Contact
ctr-contact@cspc.cn
0311-69085587
LIN
Contact

Oversight

Data monitoring committee
No
FDA-regulated drug
No
FDA-regulated device
No
View the source record on ClinicalTrials.gov ↗

Not currently enrolling

This study is not yet recruiting, as verified in Jul 2026. You cannot join it, but the record below documents what was studied.

Follow this study

Get an email when the registry record changes — status, dates, results — or when someone posts here.

Sign in to follow

Discussion

Questions and observations about this study, from anyone following it. Not medical advice, and not a channel to the study team — their contact details are on the registry record.

Sign in to join the discussion. Reading takes no account; posting does. You choose a display name, and a pseudonym is the default.

Nothing here yet. If you are running this trial, taking part in it, or weighing whether to, this is the place to say so.

Start the discussion