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RecruitingNCT06881784RASolve 301Updated Sep 29, 2026

Study of Daraxonrasib (RMC-6236) in Patients With RAS Mutated NSCLC (RASolve 301)

A Phase 3 interventional study of daraxonrasib and docetaxel in NSCLC (Non-small Cell Lung Cancer), Non-Small Cell Lung Cancer and NSCLC, sponsored by Revolution Medicines, Inc.. Recruiting at 158 sites in 19 countries. Open to participants aged 18 Years and older. Per ClinicalTrials.gov, last updated 2026-09-29.

Sponsored by Revolution Medicines, Inc. · Phase 3, Interventional, and Treatment

Phase
Phase 3
Study type
Interventional
Enrollment
590
Allocation
Randomized
Ages
18 Years and older
Sex
All
01

Study summary

The purpose of this study is to evaluate the safety and efficacy of a novel RAS(ON) inhibitor compared to docetaxel.

Read the detailed description

This is a global, randomized, open-label, Phase 3 study designed to evaluate whether treatment with daraxonrasib will improve progression free survival (PFS) or overall survival (OS) compared to docetaxel chemotherapy in patients with NSCLC who were previously treated. Patients will be randomized in a 1:1 ratio to receive daraxonrasib or docetaxel chemotherapy.

02

Conditions studied

  • NSCLC (Non-small Cell Lung Cancer)
  • Non-Small Cell Lung Cancer
  • NSCLC
  • NSCLC (Non-small Cell Lung Carcinoma)
  • NSCLC (Advanced Non-small Cell Lung Cancer)

Keywords

  • NSCLC
  • Non-Small Cell Lung Cancer
  • Lung Cancer
  • RAS
  • KRAS
  • HRAS
  • NRAS
  • RAS Q61 Mutation
  • RAS G12 Mutation
  • RAS G13 Mutation
03

Who can participate

Ages eligible
18 Years and older
Sexes eligible
All
Accepts healthy volunteers
No

Inclusion criteria

  • At least 18 years old and has provided informed consent.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
  • Pathologically confirmed NSCLC, either locally advanced or metastatic, not amenable to curative surgery or radiotherapy.
  • Measurable disease per RECIST v1.1.
  • Adequate organ function (bone marrow, liver, kidney, coagulation).
  • One to two prior lines of therapy including an anti-PD-1/anti-PD(L)-1 agent and platinum-based chemotherapy.
  • Documented RAS mutation status, defined as Nonsynonymous mutations in KRAS, NRAS, or HRAS at codons 12, 13, or 61 (G12, G13, or Q61).
  • Able to take oral medications.

Exclusion criteria

Exclusion Criteria:

  • Prior therapy with direct RAS-targeted therapy or docetaxel.
  • Untreated central nervous system (CNS) metastases.
  • Medically significant comorbidities (significant cardiovascular disease, lung disease, or impaired GI function).
  • Ongoing anticancer therapy.
  • Pregnant or breastfeeding.
04

Study design

Phase
Phase 3
Primary purpose
Treatment
Allocation
Randomized
Intervention model
Parallel assignment
Masking
None (open label)
Enrollment
590 participants (estimated)

Study arms

  • Experimental
    daraxonrasib

    study drug

    Drug: daraxonrasib

  • Active comparator
    docetaxel

    Patients randomized to the comparator control arm will receive docetaxel as the standard of care therapy.

    Drug: docetaxel

Interventions

  • Drugdaraxonrasib

    oral tablets

  • Drugdocetaxel

    intravenous (IV) infusion

05

What researchers measure

Primary outcomes

  1. Progression free survival (PFS) per Blinded Independent Central Review (BICR) in the RAS G12X-C population (i.e RAS G12X excluding G12C)

    PFS is defined as the time from randomization until disease progression or death from any cause, whichever occurs first. Progression is per response evaluation criteria in solid tumors (RECIST) v1.1 and as assessed by BICR.

    Time frame: Up to approximately 4 years

  2. Overall survival (OS) in the RAS G12X-C population

    OS is defined as the time from randomization until death from any cause.

    Time frame: Up to approximately 4 years

Secondary outcomes

  1. PFS in the RAS (MUT) population per BICR

    PFS is defined as time from randomization until disease progression or death from any cause, whichever occurs first. Progression is per RECIST v1.1 as assessed by BICR.

    Time frame: Up to approximately 4 years

  2. OS in the RAS (MUT) population

    OS is defined as time from randomization until death from any cause.

    Time frame: up to approximately 4 years

  3. Objective response per BICR in the RAS (G12X-C) and RAS (MUT) populations

    Objective response of partial response (PR) or complete response (CR) per RECIST v1.1 as assessed by BICR.

    Time frame: Up to approximately 4 years

  4. PFS per Investigator in the RAS (G12X-C) and RAS (MUT) populations

    PFS is defined as time from randomization until disease progression or death from any cause, whichever occurs first. Progression is per RECIST v1.1 as assessed by Investigator.

    Time frame: Up to approximately 4 years

  5. Objective response per Investigator in the RAS (G12X-C) and RAS (MUT) populations

    Objective response of PR or CR per RECIST v1.1 as assessed by Investigator.

    Time frame: Up to approximately 4 years

  6. Duration of response (DOR) per Investigator and per BICR in the RAS (G12X-C) and RAS (MUT) populations

    DOR is defined as time from first evidence of objective response (PR or CR) to disease progression or death due to any cause, whichever occurs first, as assessed by Investigator and by BICR.

    Time frame: Up to approximately 4 years

  7. Time to response (TTR) per Investigator and per BICR in the RAS (G12X-C) and RAS (MUT) populations

    TTR is defined as time from randomization to first evidence of objective response (PR or CR), as assessed by Investigator and by BICR.

    Time frame: Up to approximately 4 years

  8. Treatment effect on quality of life (QoL) using EORTC QLQ-LC13 In the RAS (G12X-C) and RAS (MUT) populations

    Time to deterioration (TTD) in selected symptoms (dyspnea, chest pain, cough) defined as the time from randomization to the first onset of 10 points or more deterioration from baseline in the corresponding symptom scales (dyspnea, chest pain, cough) on European Organisation for Research and Treatment of Cancer Quality of Life Questionnaire LC-13 (EORTC QLQ-LC13). Change from baseline on EORTC QLQ-LC13 in symptom scales (dyspnea, cough, chest pain).

    Time frame: Up to approximately 4 years

  9. Treatment effect on quality of life (QoL) using EORTC QLQ-C30 In the RAS (G12X-C) and RAS (MUT) populations

    Change from baseline in global quality of life score from European Organisation for Research and Treatment of Cancer Quality of Life Questionnaire C30 (EORTC QLQ-C30) questionnaire. Change from baseline on EORTC QLQ-C30 functioning domains (physical role, cognitive, emotional, social).

    Time frame: Up to approximately 4 years

  10. Safety and tolerability in the RAS (G12X-C) and RAS (MUT) population

    Incidence of treatment emergent adverse events (TEAEs), treatment related adverse events (TRAEs), serious adverse events (SAEs), changes in vital signs and clinical laboratory tests.

    Time frame: Up to approximately 4 years

  11. PK characterization of daraxonrasib In the RAS (MUT) population

    Predose and post-dose blood concentrations of daraxonrasib over time.

    Time frame: Up to approximately 4 years

06

Study locations

158 of 158 sites recruiting
  • Alabama Oncology
    Birmingham, Alabama 35243, United States
    Recruiting
  • MemorialCare Long Beach Medical Center
    Long Beach, California 90806, United States
    Recruiting
  • Yale University, Smillow Cancer Center
    New Haven, Connecticut 06519, United States
    Recruiting
  • Florida Cancer Specialists & Research Institute - South
    Fort Myers, Florida 33901, United States
    Recruiting
  • BRCR Global
    Plantation, Florida 33322, United States
    Recruiting
  • Cancer Care Centers of Breevard
    Rockledge, Florida 32955, United States
    Recruiting
  • Florida Cancer Specialists & Research Institute - North
    St. Petersburg, Florida 33705, United States
    Recruiting
  • Cleveland Clinic Martin North
    Stuart, Florida 34994, United States
    Recruiting
  • Florida Cancer Specialists & Research Institute - East
    West Palm Beach, Florida 33401, United States
    Recruiting
  • University Cancer and Blood Center
    Athens, Georgia 30607, United States
    Recruiting
  • Piedmont Healthcare, Inc
    Atlanta, Georgia 30318, United States
    Recruiting
  • Winship Cancer Institute
    Atlanta, Georgia 30322, United States
    Recruiting
  • University of Illinois Cancer Center
    Chicago, Illinois 60612, United States
    Recruiting
  • Center for Care and Discovery
    Chicago, Illinois 60637, United States
    Recruiting
  • University of Iowa Health Care Cancer Services Quad Cities
    Bettendorf, Iowa 52722, United States
    Recruiting
  • University of Iowa Hospitals & Clinics
    Iowa City, Iowa 52242, United States
    Recruiting
  • University of Iowa Health Care, Mission Cancer + Blood
    Waukee, Iowa 50263, United States
    Recruiting
  • The University of Kansas Cancer Center
    Westwood, Kansas 66205, United States
    Recruiting
  • Johns Hopkins University of Medicine
    Baltimore, Maryland 21224, United States
    Recruiting
  • Trinity Health Ann Arbor Hospital
    Ann Arbor, Michigan 48106, United States
    Recruiting
  • Karmanos Cancer Institute
    Detroit, Michigan 48201, United States
    Recruiting
  • Henry Ford Health
    Detroit, Michigan 48202, United States
    Recruiting
  • Washington University School of Medicine - Siteman Cancer Center
    St Louis, Missouri 63110, United States
    Recruiting
  • St. Vincent Frontier Cancer Center
    Billings, Montana 59102, United States
    Recruiting
  • Dartmouth-Hitchcock Medical Center
    Lebanon, New Hampshire 03756, United States
    Recruiting
  • John Theurer Cancer Center at Hackensack UMC
    Hackensack, New Jersey 07601, United States
    Recruiting
  • Morristown Medical Center (MMCORC)
    Morristown, New Jersey 07960, United States
    Recruiting
  • Roswell Park Cancer Institute
    Buffalo, New York 14263, United States
    Recruiting
  • Memorial Sloan Kettering Cancer Center
    New York, New York 10065, United States
    Recruiting
  • Montefiore Medical Center
    The Bronx, New York 10461, United States
    Recruiting
  • UNC Lineberger Comprehensive Cancer Center at University of North Carolina
    Chapel Hill, North Carolina 27599, United States
    Recruiting
  • TriHealth Cancer & Blood Institute Research
    Cincinnati, Ohio 45220, United States
    Recruiting
  • Taylor Cancer Research Center
    Maumee, Ohio 43537, United States
    Recruiting
  • Oncology Associates of Oregon PC
    Eugene, Oregon 97401, United States
    Recruiting
  • Penn State Milton S. Hershey Medical Center
    Hershey, Pennsylvania 17033, United States
    Recruiting
  • Avera Saint Luke's Hospital
    Aberdeen, South Dakota 57401, United States
    Recruiting
  • Avera Cancer Institute
    Sioux Falls, South Dakota 57105, United States
    Recruiting
  • SCRI Oncology Partners - Tennessee
    Nashville, Tennessee 37203, United States
    Recruiting
  • Texas Oncology - South Austin
    Austin, Texas 78745, United States
    Recruiting
  • Texas Oncology Dallas
    Dallas, Texas 75251, United States
    Recruiting
  • MD Anderson Cancer Center
    Houston, Texas 77030, United States
    Recruiting
  • Texas Oncology - Gulf Coast
    The Woodlands, Texas 77380, United States
    Recruiting
  • Utah Cancer Specialists
    Salt Lake City, Utah 84106, United States
    Recruiting
  • Huntsman Cancer Institute
    Salt Lake City, Utah 84112, United States
    Recruiting
  • Virginia Cancer Specialists
    Fairfax, Virginia 22031, United States
    Recruiting
  • Blacktown Medical Oncology Research, Blacktown Hospital
    Blacktown, New South Wales 2148, Australia
    • Bo Gao · Contact · 02 9881 8000
    Recruiting
  • Blacktown Medical Oncology Research
    Blacktown, New South Wales 2148, Australia
    Recruiting
  • Chris O'Brien Lifehouse
    Camperdown, New South Wales 2050, Australia
    Recruiting
  • St. George Private Hospital Clinical Trials Unit
    Kogarah, New South Wales 2217, Australia
    Recruiting
  • Calvary Mater Newcastle
    Waratah, New South Wales 2298, Australia
    Recruiting
  • Mater Misericordiae Limited
    South Brisbane, Queensland 4101, Australia
    Recruiting
  • Alfred House
    Melbourne, Victoria 3004, Australia
    Recruiting
  • Sir Charles Gairdner Hospital
    Perth, Western Australia 6009, Australia
    Recruiting
  • Institut Jules Bordet
    Anderlecht, Belgium 1070, Belgium
    Recruiting
  • Grand Hôpital de Charleroi - Les Viviers
    Gilly, 6060, Belgium
    Recruiting
  • AZ Groeninge
    Kortrijk, 8500, Belgium
    Recruiting
  • UZ Leuven-Campus Gasthuisberg
    Leuven, 3000, Belgium
    Recruiting
  • AZ Delta
    Roeselare, 8800, Belgium
    Recruiting
  • CHU Strasbourg - Nouvel Hôpital Civil
    Strasbourg, Bas Rhin 67091, France
    Recruiting
  • Hopital Nord - CHU Marseille
    Marseille, Bouches-du-Rhône 13915, France
    Recruiting
  • Institut régional du Cancer de Montpellier
    Montpellier, Herault 34298, France
    Recruiting
  • CHU Rennes Hôpital Pontchaillou
    Rennes, Ille et Vilaine 35033, France
    Recruiting
  • CHU de Grenoble - Hôpital Albert Michallon
    La Tronche, Isere 38700, France
    Recruiting
  • CHU Nantes - Hôpital Guillaume et René Laënnec
    Saint-Herblain, Loire Atlantique 44805, France
    Recruiting
  • Institut de Cancerologie de l Ouest
    Saint-Herblain, Loire Atlantique 44805, France
    Recruiting
  • Centre Leon Berard
    Léon, Lyon 69008, France
    Recruiting
  • Hopital Albert Calmette - CHU Lille
    Lille, Nord 59037, France
    Recruiting
  • Hôpital Bichat - Claude Bernard
    Paris, Paris 75018, France
    Recruiting
  • Hopital Louis Pradel
    Bron, Rhone 69677, France
    Recruiting
  • Centre Hospitalier Intercommunal de Créteil
    Créteil, Val de Marne 94000, France
    Recruiting
  • Institut Gustave Roussy
    Vaillant, Villejuif 94800, France
    Recruiting
  • CHU Brest - Hôpital Morvan
    Brest, 29200, France
    Recruiting
  • Institut Bergonie
    Gironde, 33076, France
    Recruiting
  • CHU de Toulouse - Hopital Larrey
    Toulouse, 31059, France
    Recruiting
  • LKI Lungenfachklinik Immenhausen
    Immenhausen, Hesse 34376, Germany
    Recruiting
  • Universitaetsklinikum Essen
    Essen, North Rhine-Westphalia 45147, Germany
    Recruiting
  • Universitaetsklinikum Carl Gustav Carus TU Dresden
    Dresden, Saxony 01307, Germany
    Recruiting
  • Thoraxklinik Heidelberg gGmbH
    Baden, Wuerttemberg 69469, Germany
    Recruiting
  • Klinikum Esslingen GmbH
    Baden, 73730, Germany
    Recruiting
  • Evangelische Lungenklinik Berlin
    Berlin, 13125, Germany
    Recruiting
  • Hong Kong United Oncology Centre
    Hong Kong, Hong Kong
    Recruiting
  • Queen Mary Hospital
    Hong Kong, Hong Kong
    Recruiting
  • Princess Margaret Hospital
    Lai Chi Kok, Hong Kong
    • Fiona Mei Ying Lim · Contact · 2990 2393
    Recruiting
  • The Chinese University of Hong Kong
    Shatin, 00000, Hong Kong
    • Molly LI · Contact · 35051042
    Recruiting
  • Cork Univeristy Hospital
    Cork, Cork T12 DC4A, Ireland
    Recruiting
  • Mater Private Hospital
    Dublin, Dublin 7, Ireland
    Recruiting
  • University Hospital Limerick
    Cork, Limerick V94 F858, Ireland
    Recruiting
  • Tallaght University Hospital
    Dublin, 24, Ireland
    Recruiting
  • Beaumont Hospital Cancer Clinical
    Dublin, D09 V2N0, Ireland
    Recruiting
  • Galway University Hospital
    Galway, H91 YR71, Ireland
    Recruiting
  • IEO Istituto Europeo di Oncologia
    Milan, Milano 20141, Italy
    Recruiting
  • Azienda Socio Sanitaria Territoriale Niguarda
    Milan, Milano 21206, Italy
    Recruiting
  • Istituto Clinico Humanitas
    Rossano, Milano 20089, Italy
    Recruiting
  • Fondazione IRCCS San Gerardo dei Tintori
    Monza, Milan 20900, Italy
    • Diego Luigi Cortinovis · Contact · diegoluigi.cortinovis@irccs-sa
    Recruiting
  • Istituto Nazionale Tumori Fondazione G. Pascale
    Naples, Napoli 80131, Italy
    Recruiting
  • Azienda Ospedaliero Universitaria Pisana (Presidio di Cisanello)
    Pisa, Pisa 56124, Italy
    Recruiting
  • Istituto Nazionale dei Tumori Regina Elena IRCCS
    Roma, Roma 00144, Italy
    Recruiting
  • Fondazione Policlinico Universitario Agostino Gemelli IRCCS
    Rome, 00168, Italy
    Recruiting
  • Aichi Cancer Center Hospital
    Nagoya, Aichi-ken 464-8681, Japan
    • · Contact · 052-762-6111
    Recruiting
  • Fujita Health University Hospital
    Toyoake-shi, Aichi-ken 470-1192, Japan
    • · Contact · 0562-93-2111
    Recruiting

Showing the first 100 of 158 sites across 19 countries.

07

Registry details

Key details

Study ID
NCT06881784
Lead sponsor
Revolution Medicines, Inc.
Responsible party
Sponsor
First posted
Mar 18, 2025
Start date
May 6, 2025
Primary completion
Dec 1, 2027 (estimated)
Completion
Dec 1, 2030 (estimated)
Last update
Sep 29, 2026

Study contacts

Revolution Medicines Study Director
Contact
medinfo@revmed.com
1-844-2-REVMED

Oversight

Data monitoring committee
Yes
FDA-regulated drug
Yes
FDA-regulated device
No
View the source record on ClinicalTrials.gov ↗

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