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RecruitingNCT04098744ART-CIN_IIBUpdated Oct 2, 2025

Artesunate Vaginal Inserts for the Treatment of Cervical Intraepithelial Neoplasia (CIN2/3)

A Phase 2 interventional study of Artesunate vaginal insert and Placebo vaginal insert in CIN 2/3, HPV Infection and Pre-Cancerous Dysplasia, sponsored by Frantz Viral Therapeutics, LLC. Recruiting at 7 sites in United States. Open to female participants aged 25 Years to 100 Years. Per ClinicalTrials.gov, last updated 2025-10-02.

Sponsored by Frantz Viral Therapeutics, LLC · Phase 2, Interventional, and Treatment

Phase
Phase 2
Study type
Interventional
Enrollment
78
Allocation
Randomized
Ages
25 Years to 100 Years
Sex
Female
01

Study summary

This is a phase II double blind, placebo-controlled, randomized study of Artesunate vaginal inserts for the treatment of women who have cervical high grade intraepithelial neoplasia (CIN2/3).

Read the detailed description

Eligible participants in this study are randomized 2:1 to receive either artesunate or placebo vaginal inserts for the treatment of CIN2/3. Both groups receive three 5-day cycles of the respective drug, at weeks 0, 2, and 4. Dosing visits can be done as telehealth visits (medication is mailed to the patient's home). Participants are followed after receiving artesunate at weeks 6, 17, and 40. All participants undergo a LEEP procedure at week 17.

Primary Objective: To evaluate the histopathologic response to three 5-day cycles of artesunate vaginal inserts in adult females with biopsy-proven HPV-associated CIN 2/3.

Secondary Objectives:

  • To evaluate the safety of artesunate vaginal inserts for the treatment of CIN2/3
  • To evaluate the viral clearance after three 5-day cycles of artesunate vaginal inserts in adult females with biopsy-proven HPV-associated CIN 2/3.
  • To evaluate viral clearance after three 5-day cycles of artesunate and the LEEP procedure
02

Conditions studied

  • CIN 2/3
  • HPV Infection
  • Pre-Cancerous Dysplasia
  • Cervical Dysplasia
  • HPV Related Disease

Keywords

  • treatment study
  • cancer prevention
  • non-surgical
  • HPV related disease
  • CIN
  • topical treatment
  • vaginal inserts
  • artesunate
  • artemisinin
  • non-invasive
  • high risk HPV
  • vaginal suppository
03

Who can participate

Ages eligible
25 Years to 100 Years
Sexes eligible
Female
Accepts healthy volunteers
No

Inclusion criteria

  • Adult females age ≥ 25 years
  • Capable of informed consent
  • Any HPV genotype detectable by DNA test/HPV genotyping
  • Colposcopically-directed, histologically confirmed tissue diagnosis of cervical high grade squamous intraepithelial lesions (CIN2, CIN3, or CIN2/3)
  • Women of childbearing potential agree to use birth control through week17 of the study.
  • Weight ≥ 50kg

Exclusion criteria

Exclusion Criteria:

  • Pregnant and nursing women
  • Active autoimmune disease
  • Taking immunosuppressive medication
  • HIV seropositivity
  • Immunocompromised subjects
  • Evidence of concurrent cervical adenocarcinoma in situ
  • Concurrent malignancy except for nonmelanoma skin lesions, because treatment for other cancers have systemic effects
04

Study design

Phase
Phase 2
Primary purpose
Treatment
Allocation
Randomized
Intervention model
Parallel assignment
Masking
Double (Participant, Investigator)
Enrollment
78 participants (estimated)

Study arms

  • Experimental
    Artesunate vaginal insert

    Participants will receive three 5-day cycles of artesunate vaginal inserts, 200mg/day, at week 0, week 2, week 4.

    Drug: Artesunate vaginal insert

  • Placebo comparator
    Placebo vaginal inserts

    Participants will receive three 5-day cycles of placebo vaginal inserts, at week 0, week 2, and week 4.

    Drug: Placebo vaginal insert

Interventions

  • DrugArtesunate vaginal insert

    Artesunate formulated as vaginal inserts, 200mg

    Also known as: Artesunic acid, DHA, artemisinin

  • DrugPlacebo vaginal insert

    Placebo for artesunate vaginal inserts

05

What researchers measure

Primary outcomes

  1. Proportion of participants with histologic regression by week 17

    Number of participants who undergo histologic regression to cervical intraepithelial neoplasia (CIN) 1 or less by week 17, following three 5-day cycles of artesunate vaginal inserts, as determined by the LEEP histopathologic analysis

    Time frame: 17 weeks

Secondary outcomes

  1. Number of participants who have achieved clearance of detectable human papilloma virus (HPV) by week 17

    Number of participants who had HPV strains detected at study entry which become undetectable by week 17

    Time frame: 17 weeks

  2. Number of participants who have achieved clearance of detectable human papilloma virus (HPV) after three 5-day cycles of artesunate and the LEEP procedure.

    Number of participants who had HPV strains detected at study entry which become undetectable after three 5-day cycles of artesunate and the LEEP procedure

    Time frame: 40 weeks

Other outcomes

  1. Number of participants with Treatment-Emergent Adverse Events (TEAE)

    Number of participants who had adverse events, as defined by CTCAE v5.0, related to the study intervention

    Time frame: 6 weeks

  2. Number of participants who withdrew from the study due to TEAEs

    Number of participants who were withdrawn from the study due to adverse events related to the study drug

    Time frame: 6 weeks

06

Study locations

7 of 7 sites recruiting
  • Florida Gynecologic Oncology
    Fort Myers, Florida 33905, United States
    • Cami Hansen · Contact · cami.hansen25@gmail.com · 239-334-6626
    • Fadi Abu Shahin, MD · Principal investigator
    • Samith Sandadi, MD · Sub investigator
    Recruiting
  • University of Michigan
    Ann Arbor, Michigan 48109, United States
    • Mubeenah Syedah · Contact · symubeen@med.umich.edu · 734-998-6349
    • Diane Harper, MD · Principal investigator
    Recruiting
  • Cleveland Clinic Fairview Hospital
    Cleveland, Ohio 44111, United States
    • Donna White · Contact · whited11@ccf.org · 216-445-8090
    • Megan Park · Contact · parkm2@ccf.org · 216-445-8090
    • Chad Michener, MD · Principal investigator
    • Mariam AlHilli, MD · Sub investigator
    • Steven Waggonner, MD · Sub investigator
    • Robert DeBernardo, MD · Sub investigator
    • Roberto Vargas, MD · Sub investigator
    Recruiting
  • Cleveland Clinic Foundation
    Cleveland, Ohio 44195, United States
    • Donna White · Contact · whited11@ccf.org · 216-445-8090
    • Megan Park · Contact · parkm2@ccf.org · 216-445-8090
    • Chad Michener, MD · Principal investigator
    • Mariam AlHilli, MD · Sub investigator
    • Steven Waggonner, MD · Sub investigator
    • Robert DeBernardo, MD · Sub investigator
    • Roberto Vargas, MD · Sub investigator
    Recruiting
  • Hillcrest Hospital
    Mayfield Heights, Ohio 44124, United States
    • Donna White · Contact · whited11@ccf.org · 216-445-8090
    • Megan Park · Contact · parkm2@ccf.org · 216-445-8090
    • Chad Michener, MD · Principal investigator
    • Mariam AlHilli, MD · Sub investigator
    • Steven Waggonner, MD · Sub investigator
    • Robert DeBernardo, MD · Sub investigator
    • Roberto Vargas, MD · Sub investigator
    • Lindsey Beffa, MD · Sub investigator
    Recruiting
  • The Harris Health System (L.B.J Hospital)
    Houston, Texas 77026, United States
    Recruiting
  • University of Texas, M.D. Anderson
    Houston, Texas 77030, United States
    Recruiting
07

References and documents

Individual participant data

Plan to share: No

No publications or documents are linked to this record.

08

Registry details

Key details

Study ID
NCT04098744
Lead sponsor
Frantz Viral Therapeutics, LLC
Collaborators
Amarex Clinical Research, M.D. Anderson Cancer Center, Harris Health System (L.B.J. Hospital), The Cleveland Clinic, University of Michigan, Florida Gynecologic Oncology
Responsible party
Sponsor
First posted
Sep 23, 2019
Start date
Sep 9, 2020
Primary completion
Jul 31, 2026 (estimated)
Completion
Dec 31, 2026 (estimated)
Last update
Oct 2, 2025

Study contacts

Mihaela Plesa, BA, CCRP
Contact
FVTinfo@frantzgroup.com
440-255-1155 ext. 100
Ahmad Bayat, MD
Contact
ahmadb@amarexcro.com
(301) 956-2523

Oversight

Data monitoring committee
Yes
FDA-regulated drug
Yes
FDA-regulated device
No
View the source record on ClinicalTrials.gov ↗

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